Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Protein mono-ADP-ribosyltransferase TIPARP' and Ligand = 'BDBM431024'
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Ribon Therapeutics Inc.

US Patent
LigandPNGBDBM431024(5-[6-(piperidin-4-yloxy)-1H,2H,3H-pyrrolo[3,4-c]py...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Displacement of Probe A, a biotinylated probe binding to the TIPARP active site, was measured using a time-resolved fluorescence energy transfer (TR-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JM2D1ZUS Patent
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Ribon Therapeutics Inc.

US Patent
LigandPNGBDBM431024(5-[6-(piperidin-4-yloxy)-1H,2H,3H-pyrrolo[3,4-c]py...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Displacement of Probe A, a biotinylated probe binding to the TIPARP active site, was measured using a time-resolved fluorescence energy transfer (TR-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69NPPUS Patent
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Ribon Therapeutics Inc.

US Patent
LigandPNGBDBM431024(5-[6-(piperidin-4-yloxy)-1H,2H,3H-pyrrolo[3,4-c]py...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Displacement of Probe A, a biotinylated probe binding to the TIPARP active site, was measured using a time-resolved fluorescence energy transfer (TR-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VQ35S4US Patent