Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Protein-glutamine gamma-glutamyltransferase 6' and Ligand = 'BDBM185173'
TargetProtein-glutamine gamma-glutamyltransferase 6(Homo sapiens (Human))
Aston University

LigandPNGBDBM185173(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222SJCPubMed