Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Protein-glutamine gamma-glutamyltransferase K' and Ligand = 'BDBM185176'
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Aston University

LigandPNGBDBM185176([2-[[2-[4-(1-Adamantylmethoxycarbonyl)piperazin-1-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222SJCPubMed