Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Protein-serine O-palmitoleoyltransferase porcupine' and Ligand = 'BDBM50133866'
TargetProtein-serine O-palmitoleoyltransferase porcupine(Homo sapiens (Human))
Experimental Therapeutics Centre

Curated by ChEMBL
LigandPNGBDBM50133866(CHEMBL3633802)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Inhibition of porcupine in human HEK293 cells assessed as reduction in Wnt secretion by measuring suppression of beta-catenin reporter activity after...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21838C2PubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Homo sapiens (Human))
Experimental Therapeutics Centre

Curated by ChEMBL
LigandPNGBDBM50133866(CHEMBL3633802)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Inhibition of porcupine (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FF5PubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Mus musculus)
Experimental Therapeutics Centre

Curated by ChEMBL
LigandPNGBDBM50133866(CHEMBL3633802)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of mouse porcupine expressed in human HT1080 cells assessed as reduction in beta catenin reporter activity using firefly luciferase substr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21838C2PubMed