Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Proteinase-activated receptor 1' and Ligand = 'BDBM50079754'
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Oregon Health& Science University

Curated by ChEMBL
LigandPNGBDBM50079754(CHEMBL65476 | N*3*-Cyclopropyl-7-(4-isopropyl-benz...)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Antagonist activity at PAR1 in human platelet membranes assessed as inhibition of interaction of PAR1 with [Ala-Phe(p-F)-Arg-Cha-HArg-Tyr-NH2] by Chr...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QN68NSPubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Oregon Health& Science University

Curated by ChEMBL
LigandPNGBDBM50079754(CHEMBL65476 | N*3*-Cyclopropyl-7-(4-isopropyl-benz...)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Inhibitory activity against binding to Thrombin receptor 1 (PAR-1)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25X284BPubMed