Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Proto-oncogene tyrosine-protein kinase Src' and Ligand = 'BDBM50184780'
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50184780(CHEMBL3823255 | US10294227, Code 526)copy SMILEScopy InChI
Affinity DataIC50: 114nMAssay Description:Inhibition of C-terminal His-tagged full length human SRC expressed in insect cells preincubated for 20 mins using poly[Glu,Tyr]4:1 as substrate meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85B2DPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50184780(CHEMBL3823255 | US10294227, Code 526)copy SMILEScopy InChI
Affinity DataIC50: 550nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27D2XFPUS Patent