Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Proto-oncogene tyrosine-protein kinase Src' and Ligand = 'BDBM50389679'
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389679(CHEMBL2070046 | US10544104, Compound 135 | US97650...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human SRC using Ac-EIYGEFKKK-OH as substrate after 60 mins by phosphorimaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2706VPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389679(CHEMBL2070046 | US10544104, Compound 135 | US97650...)copy SMILEScopy InChI
Affinity DataIC50: 2.01E+3nMAssay Description:Inhibition of TgCDPK1 and CpCDPK1 was determined using a luminescent kinase assay which measures ATP depletion in the presence of the Syntide 2 pepti...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D79DSFUS Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50389679(CHEMBL2070046 | US10544104, Compound 135 | US97650...)copy SMILEScopy InChI
Affinity DataIC50: 2.01E+3nMAssay Description:Inhibition of human tyrosine kinases.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B56MVCUS Patent