Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Pyroglutamylated RF-amide peptide receptor' and Ligand = 'BDBM50396416'
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50396416(CHEMBL2170398)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as inhibition of human 26RFa-induced increase in intracell...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VSGPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50396416(CHEMBL2170398)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VSGPubMed