Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Pyroglutamylated RF-amide peptide receptor' and Ligand = 'BDBM50396420'
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50396420(CHEMBL2170390)copy SMILEScopy InChI
Affinity DataIC50: 2.99E+3nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VSGPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50396420(CHEMBL2170390)copy SMILEScopy InChI
Affinity DataEC50:  136nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VSGPubMed