Found 2 Enz. Inhib. hit(s) with Target = 'Pyroglutamylated RF-amide peptide receptor' and Ligand = 'BDBM50396420'
Affinity DataIC50: 2.99E+3nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
Affinity DataEC50: 136nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair