Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Pyroglutamylated RF-amide peptide receptor' and Ligand = 'BDBM50469430'
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Normandy University

Curated by ChEMBL
LigandPNGBDBM50469430(CHEMBL4279100)copy SMILEScopy InChI
Affinity DataIC50: 8.25E+3nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Normandy University

Curated by ChEMBL
LigandPNGBDBM50469430(CHEMBL4279100)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as increase Ca2+ mobilization after 3 mins by Fluo-4 AM-based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed