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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'RAC-alpha serine/threonine-protein kinase' and Ligand = 'BDBM130222'
Target
RAC-alpha serine/threonine-protein kinase
(Homo sapiens (Human))
ArQule, Inc.
US Patent
Ligand
BDBM130222
(US8815854, 11)
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Affinity Data
IC50: 1.99nM
pH: 8.0
Assay Description:
AKT1 activity was assayed using the GSK3-derived biotinylated peptide substrate, crosstide (biotin-GRPRTSSFAEG), and AlphaScreen (Amplified Luminesce...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2J67FMR
US Patent