Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'RAC-alpha serine/threonine-protein kinase' and Ligand = 'BDBM130222'
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
ArQule, Inc.

US Patent
LigandPNGBDBM130222(US8815854, 11)copy SMILEScopy InChI
Affinity DataIC50: 1.99nMpH: 8.0Assay Description:AKT1 activity was assayed using the GSK3-derived biotinylated peptide substrate, crosstide (biotin-GRPRTSSFAEG), and AlphaScreen (Amplified Luminesce...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J67FMRUS Patent