Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'RAC-alpha serine/threonine-protein kinase' and Ligand = 'BDBM180366'
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
SANOFI

US Patent
LigandPNGBDBM180366(US9133168, Example 21c | US9133168, Example 22c)copy SMILES
Affinity DataIC50: 2nMAssay Description:This test is based on measurement of the expression of AKT protein phosphorylated on serine 473 (P-AKT-S473) in the PC3 human prostate carcinoma line...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29W0D8XUS Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
SANOFI

US Patent
LigandPNGBDBM180366(US9133168, Example 21c | US9133168, Example 22c)copy SMILES
Affinity DataIC50: 17nMAssay Description:This test is based on measurement of the expression of AKT protein phosphorylated on serine 473 (P-AKT-S473) in the PC3 human prostate carcinoma line...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29W0D8XUS Patent