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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'RAC-alpha serine/threonine-protein kinase' and Ligand = 'BDBM24841'
Target
RAC-alpha serine/threonine-protein kinase
(Homo sapiens (Human))
Pfizer
Ligand
BDBM24841
(N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-7H-py...)
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Affinity Data
IC50: 151nM
pH: 7.5 T: 2°C
Assay Description:
A fluorescence polarization IMAP type assay is used. After a 90 min incubation of reaction mixtures containing enzyme, substrate, and inhibitor, IMAP...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
DrugBank
MMDB
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M043QC
PubMed
PDB
3D Structure (crystal)