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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'RAC-alpha serine/threonine-protein kinase' and Ligand = 'BDBM50312924'
Target
RAC-alpha serine/threonine-protein kinase
(Homo sapiens (Human))
Amgen Inc.
Curated by
ChEMBL
Ligand
BDBM50312924
((S)-N1-(3-(isoquinolin-6-yl)isoxazol-5-yl)-3-(4-(t...)
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Affinity Data
IC50: 17nM
Assay Description:
Inhibition of human AKT1 in human U87MG cells assessed as PRAS40 phosphorylation after 1 hr by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
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Ligand Info
CHEMBL
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PC sid
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In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q20C4VWX
PubMed