Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Rap guanine nucleotide exchange factor 4' and Ligand = 'BDBM50175100'
TargetRap guanine nucleotide exchange factor 4(Homo sapiens (Human))
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50175100(CHEMBL3809121)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of 8-NBD-cAMP binding to EPAC2 (unknown origin) by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6335PubMed
TargetRap guanine nucleotide exchange factor 4(Homo sapiens (Human))
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50175100(CHEMBL3809121)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of EPAC2 (unknown origin) assessed as reduction in cAMP-mediated guanine nucleotide exchange factor activity in presence of C-terminal tru...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6335PubMed