Found 2 Enz. Inhib. hit(s) with Target = 'Receptor tyrosine-protein kinase erbB-2' and Ligand = 'BDBM4583' TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University of South China
Curated by ChEMBL
University of South China
Curated by ChEMBL
Affinity DataIC50: 301nMAssay Description:Inhibition of recombinant human His6-tagged HER2 cytoplasmic domain (676 to 1245 residues) expressed in baculovirus infected Sf9 insect cells assesse...More data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University of South China
Curated by ChEMBL
University of South China
Curated by ChEMBL
Affinity DataIC50: 301nMAssay Description:The HER-2 kinase autophosphorylation activity was measured by DELFIA/time-resolved fluorometry with excitation at 340 nm and emission at 615 nm. Po...More data for this Ligand-Target Pair
