Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor RXR-alpha' and Ligand = 'BDBM50143823'
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50143823((E)-3-[5-Methyl-4-(5,5,8,8-tetramethyl-5,6,7,8-tet...)copy SMILEScopy InChI
Affinity DataKi:  158nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MRCPubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50143823((E)-3-[5-Methyl-4-(5,5,8,8-tetramethyl-5,6,7,8-tet...)copy SMILEScopy InChI
Affinity DataEC50:  106nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MRCPubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50143823((E)-3-[5-Methyl-4-(5,5,8,8-tetramethyl-5,6,7,8-tet...)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+3nMAssay Description:Effective concentration for lipogenesis induced by retinoid X receptor alpha in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MRCPubMed