Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor beta' and Ligand = 'BDBM50526314'
TargetRetinoic acid receptor beta(Homo sapiens (Human))
King''s College London

US Patent
LigandPNGBDBM50526314(CHEMBL4459692 | US10752616, Code No. BHBA-001)copy SMILEScopy InChI
Affinity DataEC50:  1.94nMAssay Description:Transcriptional transactivation assays were performed with gal4 fusion receptor constructs, created using each of the RAR ligand binding domains of e...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B85C6MUS Patent
TargetRetinoic acid receptor beta(Mus musculus)
King's College

Curated by ChEMBL
LigandPNGBDBM50526314(CHEMBL4459692 | US10752616, Code No. BHBA-001)copy SMILEScopy InChI
Affinity DataEC50:  1.90nMAssay Description:Transactivation of GAL4-fused mouse RARbeta-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25142NCPubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
King''s College London

US Patent
LigandPNGBDBM50526314(CHEMBL4459692 | US10752616, Code No. BHBA-001)copy SMILEScopy InChI
Affinity DataEC50:  2.10nMAssay Description:Transactivation of GAL4 DBD-fused human RARbeta-LBD expressed in HEK293 cells by beta-lactamase reporter gene based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25142NCPubMed