Compile Data Set for Download or QSAR
Found 6 Enz. Inhib. hit(s) with Target = 'Rho-associated protein kinase 2' and Ligand = 'BDBM412136'
TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM412136(US10392402, Compound A | US10738007, Compound A | ...)copy SMILEScopy InChI
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TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM412136(US10392402, Compound A | US10738007, Compound A | ...)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
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TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM412136(US10392402, Compound A | US10738007, Compound A | ...)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMAssay Description:n general, kinases regulate many important cellular activities including cell growth, signaling, metabolism, etc. Different kinases have distinct fun...More data for this Ligand-Target Pair
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BindingDB Entry DOI: 10.7270/Q2JD51P0US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM412136(US10392402, Compound A | US10738007, Compound A | ...)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
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BindingDB Entry DOI: 10.7270/Q25Q505JUS Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM412136(US10392402, Compound A | US10738007, Compound A | ...)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
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BindingDB Entry DOI: 10.7270/Q23X890MUS Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM412136(US10392402, Compound A | US10738007, Compound A | ...)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMMore data for this Ligand-Target Pair
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BindingDB Entry DOI: 10.7270/Q22Z18MNUS Patent