Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Rhodopsin kinase GRK1' and Ligand = 'BDBM50173314'
TargetRhodopsin kinase GRK1(Homo sapiens (Human))
THE REGENTS OF THE UNIVERSITY OF MICHIGAN

US Patent
LigandPNGBDBM50173314(CHEMBL3808840 | US10023564, Example 16)copy SMILEScopy InChI
Affinity DataIC50: 7.10E+4nMpH: 7.0Assay Description:GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V126V5US Patent
TargetRhodopsin kinase GRK1(Homo sapiens (Human))
THE REGENTS OF THE UNIVERSITY OF MICHIGAN

US Patent
LigandPNGBDBM50173314(CHEMBL3808840 | US10023564, Example 16)copy SMILEScopy InChI
Affinity DataIC50: 7.10E+4nMAssay Description:Inhibition of GRK1 (unknown origin) using tubulin as substrate by SDS-PAGE methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12X4PubMed