Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Ribosomal protein S6 kinase alpha-3' and Ligand = 'BDBM50360282'
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360282(CHEMBL1933143 | US9150577, 193)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of RSK2 phosphorylation by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360282(CHEMBL1933143 | US9150577, 193)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of human RSK2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348KTRPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360282(CHEMBL1933143 | US9150577, 193)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of human RSK2-mediated CREB phosphorylation in HLR-CREB cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348KTRPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Boehringer-Ingelheim Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50360282(CHEMBL1933143 | US9150577, 193)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of RSK2-mediated CREB phosphorylation in HeLa cells expressing luciferase reporter geneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4K7NPubMed