Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase 17B' and Ligand = 'BDBM50559221'
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559221(CHEMBL4763392)copy SMILES
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559221(CHEMBL4763392)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559221(CHEMBL4763392)copy SMILES
Affinity DataKd:  910nMAssay Description:Binding affinity to N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli by KINOMEscan scan...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed