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TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Albert Einstein College of Medicine
Curated by ChEMBL
Albert Einstein College of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin) by Z'-LYTE assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Albert Einstein College of Medicine
Curated by ChEMBL
Albert Einstein College of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Albert Einstein College of Medicine
Curated by ChEMBL
Albert Einstein College of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of BRAF V600E mutant in human A375 cells assessed as reduction in ERK phosphorylation after 2 hrs by ELISAMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Albert Einstein College of Medicine
Curated by ChEMBL
Albert Einstein College of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Inhibition of wild type BRAF (unknown origin) by Z'-LYTE assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Albert Einstein College of Medicine
Curated by ChEMBL
Albert Einstein College of Medicine
Curated by ChEMBL
Affinity DataKd: 0.370nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) by KINOMEscan assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Albert Einstein College of Medicine
Curated by ChEMBL
Albert Einstein College of Medicine
Curated by ChEMBL
Affinity DataKd: 0.330nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) V600E mutant by KINOMEscan assayMore data for this Ligand-Target Pair
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