Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase Chk2' and Ligand = 'BDBM31093'
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Millennium Pharmaceuticals Inc.
Curated by ChEMBL
Millennium Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of CHK2 by radioactive flashplate assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Millennium Pharmaceuticals Inc.
Curated by ChEMBL
Millennium Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CHEK2 kinase domainMore data for this Ligand-Target Pair