Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase D1' and Ligand = 'BDBM50324339'
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50324339(3-Amino-2''-cyclohexylamino-3,4,5,6-tetrahydro-2H-...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of PKD1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84C2JPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50324339(3-Amino-2''-cyclohexylamino-3,4,5,6-tetrahydro-2H-...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Inhibition of PKD1 assessed as inhibition of HDAC5 neuclear exportMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84C2JPubMed