Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase Sgk1' and Ligand = 'BDBM50043017'
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
Dart Neuroscience LLC
Curated by ChEMBL
Dart Neuroscience LLC
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair