Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase Sgk1' and Ligand = 'BDBM50043019'
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))TBA
LigandPNGBDBM50043019(CHEMBL3355029)copy SMILES
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human SGK1 expressed in baculovirus expression system using 5-carboxyfluorescein -RPRAATF-NH2 as substrate preincubated for...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55SCWPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))TBA
LigandPNGBDBM50043019(CHEMBL3355029)copy SMILES
Affinity DataIC50: 1.5nMAssay Description:Inhibition of SGK1 (unknown origin) assessed as substrate phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))TBA
LigandPNGBDBM50043019(CHEMBL3355029)copy SMILES
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human SGK1 expressed in baculovirus expression system using 5-carboxyfluorescein -RPRAATF-NH2 as substrate preincubated for...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55SCWPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))TBA
LigandPNGBDBM50043019(CHEMBL3355029)copy SMILES
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant SGK1 (unknown origin) expressed in U2OS cells by cellular activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BFBPubMed
TargetSerine/threonine-protein kinase Sgk1(Mus musculus (Mouse))TBA
LigandPNGBDBM50043019(CHEMBL3355029)copy SMILES
Affinity DataIC50: 253nMAssay Description:Inhibition of mouse SGK1 in presence 500 uM presence of ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55SCWPubMed