Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase TBK1' and Ligand = 'BDBM357905'
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM357905(2-Amino-7-isobutyl-5-oxo-5H-chromeno[2,3-b]pyridin...)copy SMILEScopy InChI
Affinity DataIC50: 550nMAssay Description:Inhibition of human TBK1 (1 to 657 residues) expressed in Baculovirus infected SF9 insect cells using myelin basic protein as substrate in presence o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M04858PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM357905(2-Amino-7-isobutyl-5-oxo-5H-chromeno[2,3-b]pyridin...)copy SMILEScopy InChI
Affinity DataIC50: 550nMAssay Description:Inhibition of human TBK1 (1 to 657 residues) expressed in Baculovirus infected SF9 insect cells using myelin basic protein as substrate in presence o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M04858PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM357905(2-Amino-7-isobutyl-5-oxo-5H-chromeno[2,3-b]pyridin...)copy SMILEScopy InChI
Affinity DataIC50: 1.23E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N87D2SUS Patent