Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase ULK1' and Ligand = 'BDBM379444'
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
SALK INSTITUTE FOR BIOLOGICAL STUDIES; SANFORD BURNHAM PREBYS MEDICAL DISCOVERY INSTITUTE; YALE UNIVERSITY

US Patent
LigandPNGBDBM379444(6-((5-bromo-4-((4-ethyl-3,4-dihydro-2H-pyrido[3,2-...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:ULK1 inhibition assay is a screening assay to identify compounds that inhibit kinase activity of ULK1 using the ULKtide peptide. In some embodiments,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24F1TTDUS Patent
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
SALK INSTITUTE FOR BIOLOGICAL STUDIES; SANFORD BURNHAM PREBYS MEDICAL DISCOVERY INSTITUTE; YALE UNIVERSITY

US Patent
LigandPNGBDBM379444(6-((5-bromo-4-((4-ethyl-3,4-dihydro-2H-pyrido[3,2-...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Gamma-32P assays to measure ULK1 kinase activity were performed as previously described. Briefly, Flag ULK1 was transfected into HEK293T cells and 20...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N30084US Patent