Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase mTOR' and Ligand = 'BDBM174472'
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
KUDOS PHARMACEUTICALS LIMITED

US Patent
LigandPNGBDBM174472(US9102670, 4f)copy SMILEScopy InChI
Affinity DataIC50: 1.97nMAssay Description:For mTOR enzyme activity assays, mTOR protein was isolated from HeLa cell cytoplasmic extract by immunoprecipitation, and activity determined essenti...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35MZUS Patent
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
KUDOS PHARMACEUTICALS LIMITED

US Patent
LigandPNGBDBM174472(US9102670, 4f)copy SMILEScopy InChI
Affinity DataIC50: 2.70nMT: 2°CAssay Description:The assay used AlphaScreen technology (Gray et al., Analytical Biochemistry, 2003, 313: 234-245) to determine the ability of test compounds to inhibi...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35MZUS Patent