Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein phosphatase 2A activator' and Ligand = 'BDBM40776'
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66J5WPubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)copy SMILEScopy InChI
Affinity DataIC50: 7.5nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66J5WPubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66J5WPubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66J5WPubMed