Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Serine protease 1' and Ligand = 'BDBM18965'
TargetSerine protease 1(Bos taurus (bovine))
Bristol-Myers Squibb Company

LigandPNGBDBM18965(1-[3-(aminomethyl)phenyl]-3-methyl-N-[4-(2-sulfamo...)copy SMILEScopy InChI
Affinity DataKi:  248nM ΔG°:  -37.3kJ/molepH: 7.0 T: 2°CAssay Description:Ki values were obtained from purified enzyme. All assays were run in microtiter plates. Plates were read for 30 min at 405 nm. Rates were determined ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4P78PubMed
TargetSerine protease 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM18965(1-[3-(aminomethyl)phenyl]-3-methyl-N-[4-(2-sulfamo...)copy SMILEScopy InChI
Affinity DataKi:  250nMAssay Description:Tested in vitro for inhibition of human trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MP2PubMed