Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Serine protease hepsin' and Ligand = 'BDBM50272185'
TargetSerine protease hepsin(Homo sapiens (Human))
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50272185(CHEMBL4129836)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant C-terminal His10-tagged human Hepsin (R45 to L17 residues) D161E/ R162K double mutant expressed in mouse NS0 cells using Bo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3VVTPubMed
TargetSerine protease hepsin(Homo sapiens (Human))
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50272185(CHEMBL4129836)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of doxycycline induced Hepsin in human MCF10A cells using Boc-QRR-AMC as substrate preincubated for 24 hrs followed by doxycycline inducti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3VVTPubMed