Found 5 Enz. Inhib. hit(s) with Target = 'Sigma non-opioid intracellular receptor 1' and Ligand = 'BDBM50108664'
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Pharmazeutisches Institut der Universität Freiburg
Curated by ChEMBL
Pharmazeutisches Institut der Universität Freiburg
Curated by ChEMBL
Affinity DataKi: 0.690nMAssay Description:Sigma opioid receptor type 1 affinity in guinea pig brain by employing [3H](+)-pentazocine as radioligand.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut f£r Pharmazeutische und Medizinische Chemie der Westf£lischen Wilhelms-Universit£t M£nster
Curated by ChEMBL
Institut f£r Pharmazeutische und Medizinische Chemie der Westf£lischen Wilhelms-Universit£t M£nster
Curated by ChEMBL
Affinity DataKi: 0.690nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain cortex membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut f£r Pharmazeutische und Medizinische Chemie der Westf£lischen Wilhelms-Universit£t M£nster
Curated by ChEMBL
Institut f£r Pharmazeutische und Medizinische Chemie der Westf£lischen Wilhelms-Universit£t M£nster
Curated by ChEMBL
Affinity DataKi: 0.690nMAssay Description:Displacement of [3H]-pentazocine from guinea pig brain sigma 1 receptor incubated for 8 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut f£r Pharmazeutische und Medizinische Chemie der Westf£lischen Wilhelms-Universit£t M£nster
Curated by ChEMBL
Institut f£r Pharmazeutische und Medizinische Chemie der Westf£lischen Wilhelms-Universit£t M£nster
Curated by ChEMBL
Affinity DataKi: 0.690nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in Dunkin Hartley guinea pig brain membranes after 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
Pharmazeutisches Institut der Universität Freiburg
Curated by ChEMBL
Pharmazeutisches Institut der Universität Freiburg
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Sigma opioid receptor type 2 affinity in rat liver by employing [3H]ditolylguanidine as radioligandMore data for this Ligand-Target Pair