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Affinity DataKi: 0.400nMAssay Description:Displacement of [3H](+)pentazocine from sigma1 receptor in Dunkin Hartley guinea pig brain membrane after 120 mins by liquid scintillation counting a...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Universit£ di Modena and Reggio Emilia
Curated by ChEMBL
Universit£ di Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 0.490nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Universit£ di Modena and Reggio Emilia
Curated by ChEMBL
Universit£ di Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
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