Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Sodium channel protein type 9 subunit alpha' and Ligand = 'BDBM371616'
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
University of California at San Francisco

LigandPNGBDBM371616((R)-4-(2-(6-Fluoropyridin-3-yl)-4-(trifluoromethyl...)copy SMILEScopy InChI
Affinity DataIC50: 0.0400nMAssay Description:HEK-293 cells overexpressing the channel of interest were seeded in a 96-well plate at a density of 30000 cells/well and incubated at 37° C./5% CO2 f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NG4SZXUS Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
University of California at San Francisco

LigandPNGBDBM371616((R)-4-(2-(6-Fluoropyridin-3-yl)-4-(trifluoromethyl...)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Inhibition of Nav1.7 (unknown origin) expressed in HEK293 cells assessed as reduction in veratridine-induced depolarization preincubated for 15 to 20...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69P5CPubMed