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TargetSodium- and chloride-dependent GABA transporter 1(Mus musculus)
Ludwig Maximilians University at Munich
Curated by ChEMBL
Ludwig Maximilians University at Munich
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of [3H]GABA uptake at mouse GAT1 expressed in HEK293 cells after 25 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Ludwig-Maximilians-University M£nchen
Curated by ChEMBL
Ludwig-Maximilians-University M£nchen
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of GAT-1 in rat brain homogenate assessed as decrease in [3H]GABA uptake preincubated for 8 mins followed by [3H]GABA addition and measure...More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Ludwig-Maximilians-University M£nchen
Curated by ChEMBL
Ludwig-Maximilians-University M£nchen
Curated by ChEMBL
Affinity DataIC50: 148nMAssay Description:Inhibition of mouse GAT1 expressed in HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 35 mins by liquid scintillation metho...More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Ludwig-Maximilians-University M£nchen
Curated by ChEMBL
Ludwig-Maximilians-University M£nchen
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of mouse GAT1 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Ludwig-Maximilians-University M£nchen
Curated by ChEMBL
Ludwig-Maximilians-University M£nchen
Curated by ChEMBL
Affinity DataKd: 27nMAssay Description:Inhibition of NO711 binding to mouse GAT1 expressed in HEK293 cell membranes assessed as reduction in NO711 binding at incubated for 4 hrs in presenc...More data for this Ligand-Target Pair
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