Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Sodium- and chloride-dependent glycine transporter 1' and Ligand = 'BDBM50457706'
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Dart NeuroScience LLC

Curated by ChEMBL
LigandPNGBDBM50457706(CHEMBL4216391)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of GlyT1 in primary rat cortical neurons assessed as reduction in [14C]glycine uptake after 2 hrs by microbeta scintillation counting meth...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB26PMPubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Dart NeuroScience LLC

Curated by ChEMBL
LigandPNGBDBM50457706(CHEMBL4216391)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human GlyT1c expressed in HEK293 cells assessed as reduction in [14C]glycine uptake after 2 hrs by microbeta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB26PMPubMed