Found 10 Enz. Inhib. hit(s) with Target = 'Sodium-dependent dopamine transporter' and Ligand = 'BDBM50006781'
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Binding affinity to dopamine transporter (DAT) using [3H]WIN-35428 as a radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 5.80nMAssay Description:Binding affinity of compound on dopamine transporters of rat striated membranes using [3H]- mazindol.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 6.90nMAssay Description:Binding affinity for [3H]DA (Dopamine transporter) uptake by striated synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Binding affinity against Dopamine transporter using [3H]WIN-35 428 in rat striatumMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Displacement of [3H]WIN-35428 from DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of [3H]WIN-35428l binding to Dopamine transporterMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataIC50: 7.5nMAssay Description:Inhibitory activity determined for [3H]DA (Dopamine transporter) uptake by striated synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibitory activity on dopamine transporter of rat striated membranes using [3H]- mazindol.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataIC50: 23.4nMAssay Description:Displacement of [3H]WIN-35428 from DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataIC50: 23.4nMAssay Description:Displacement of [3H]WIN-35428 from DATMore data for this Ligand-Target Pair