Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Sodium-dependent noradrenaline transporter' and Ligand = 'BDBM50319597'
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Pfizer Global Research& Development

Curated by ChEMBL
LigandPNGBDBM50319597((2R)-(4-[3-(3-Methoxyphenyl)-2,2-dioxido-2,1,3-ben...)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Displacement of [3H]nisoxetine from human NET expressed in MDCK-Net6 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC32JRPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Pfizer Global Research& Development

Curated by ChEMBL
LigandPNGBDBM50319597((2R)-(4-[3-(3-Methoxyphenyl)-2,2-dioxido-2,1,3-ben...)copy SMILEScopy InChI
Affinity DataIC50: 143nMAssay Description:Inhibition of human NET-mediated norepinephrine uptake in MDCK-Net6 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC32JRPubMed