Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Solute carrier organic anion transporter family member 1A4' and Ligand = 'BDBM50375594'
TargetSolute carrier organic anion transporter family member 1A4(Rattus norvegicus)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50375594(TAUROCHOLATE)copy SMILEScopy InChI
Affinity DataKi:  3.94E+4nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp2-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XW4M2TPubMed
TargetSolute carrier organic anion transporter family member 1A4(Rattus norvegicus)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50375594(TAUROCHOLATE)copy SMILEScopy InChI
Affinity DataKi:  1.56E+5nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin uptake in Oatp2-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22N53J3PubMed
TargetSolute carrier organic anion transporter family member 1A4(Rattus norvegicus)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50375594(TAUROCHOLATE)copy SMILEScopy InChI
Affinity DataIC50: 1.48E+6nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9RQFPubMed