Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Substance-K receptor' and Ligand = 'BDBM50051291'
TargetSubstance-K receptor(Homo sapiens (Human))
SmithKline Beecham S.p.A.

Curated by ChEMBL
LigandPNGBDBM50051291(CHEMBL429951 | Phenyl-[(2-phenyl-quinoline-4-carbo...)copy SMILEScopy InChI
Affinity DataKi:  2.95E+3nMAssay Description:Binding Affinity of [125I]NKA towards Tachykinin receptor 2-CHO cell membranes (n=3-8)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6CJRPubMed
TargetSubstance-K receptor(Homo sapiens (Human))
SmithKline Beecham S.p.A.

Curated by ChEMBL
LigandPNGBDBM50051291(CHEMBL429951 | Phenyl-[(2-phenyl-quinoline-4-carbo...)copy SMILEScopy InChI
Affinity DataKi:  2.95E+3nMAssay Description:Inhibition of [125I]-Neurokinin A (NKA) binding in human Tachykinin receptor 2 of chinese hamster ovary (hNK-2-CHO) cell membranes.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6HHBPubMed