TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp& Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp& Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [125 I]Trp8-substance P displacement.More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp& Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp& Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [125 I]Trp8-substance P displacement.More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp& Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp& Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Antagonist activity at NK1 receptorMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp& Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp& Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 25.7nMAssay Description:Binding affinity was measured against the Tachykinin receptor 1 in CHO-expressed hNK1 using [125I]SP.More data for this Ligand-Target Pair