Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50066195'
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50066195((S)-1-(2-Nitro-benzylthiocarbamoyl)-pyrrolidine-2-...)copy SMILEScopy InChI
Affinity DataKi:  78nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ66QJPubMed