Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50066239'
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute for Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50066239((S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2...)copy SMILEScopy InChI
Affinity DataKi:  170nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 to displace [3H][Sar9Met(O2)11]-SP (1 nM) binding to rabbit whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ66QJPubMed