Affinity DataKi: 1.5nMAssay Description:Binding affinity of the compound for NK-1 receptor was determined in a radioligand binding assay using IM9 human lymphoblastoma cell line.More data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Antagonistic potency for NK-2 receptor was determined in vitro, using isolated rabbit pulmonary artery.More data for this Ligand-Target Pair