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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'TGF-beta receptor type-1 [T204D]' and Ligand = 'BDBM282825'
Target
TGF-beta receptor type-1 [T204D]
(Homo sapiens (Human))
University of Wisconsin at Madison
Ligand
BDBM282825
(6-(4-(3-chloro-4-fluorophenyl)-1-(2-hydroxyethyl)-...)
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Affinity Data
IC50: 1.80nM
Assay Description:
Assays for the compounds reported below were conducted in 1536-well plates and 2 mL reactions are prepared from addition of HIS-TGF-βR1 T204D or...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
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Ligand Info
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PC cid
PC sid
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In Depth
Details
BindingDB Entry DOI:
10.7270/Q2B85BFB
US Patent
PDB
3D Structure (crystal)