Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Transcription initiation factor TFIID subunit 1' and Ligand = 'BDBM50269691'
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269691(CHEMBL4076944)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed