Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = 'Transcription initiation factor TFIID subunit 1' and Ligand = 'BDBM50504160'
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)copy SMILEScopy InChI
Affinity DataKd:  5.53E+3nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: R1398-D1524More data for this Ligand-Target Pair
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)copy SMILEScopy InChI
Affinity DataKd:  17nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: D1522-D1656More data for this Ligand-Target Pair
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)copy SMILEScopy InChI
Affinity DataKd:  5.00E+3nMAssay Description:Binding affinity to TAF1 BD 1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)copy SMILEScopy InChI
Affinity DataKd:  17nMAssay Description:Binding affinity to TAF1 BD 2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)copy SMILEScopy InChI
Affinity DataKd:  147nMAssay Description:Binding affinity to human TAF1 tandem bromodomain (1373 to 1499 residues) transfected in Escherichia coli BL21 (DE3) assessed as dissociation constan...More data for this Ligand-Target Pair