Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily A member 1' and Ligand = 'BDBM191652'
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
GLENMARK PHARMACEUTICALS S.A.

US Patent
LigandPNGBDBM191652(US9186360, 51 | US9186360, 52)copy SMILEScopy InChI
Affinity DataIC50: 2.49nMT: 2°CAssay Description:The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TX3D5QUS Patent
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
GLENMARK PHARMACEUTICALS S.A.

US Patent
LigandPNGBDBM191652(US9186360, 51 | US9186360, 52)copy SMILEScopy InChI
Affinity DataIC50: 4.84nMT: 2°CAssay Description:The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TX3D5QUS Patent